Neurontin

Intended to alleviate chronic neuropathic pain and prevent seizures, utilized to support neurological stability and enhance quality of life.

Strengths: 100 · 300 · 400 · 600mg

Medicine details

Therapeutic class

Antiepileptic

Pharmacological class

GABA analogue

Known off-label uses

generalised anxiety disorder

Contraindications

hypersensitivity to gabapentin

Minor side effects

dizziness; somnolence; fatigue; nausea

Moderate side effects

peripheral oedema; ataxia; tremor

Dosage forms

Capsule, hard

Administration route

Oral use

Prescription status

POM

Manufacturer

Pfizer

Onset Time

1–2 weeks

Duration

6–8 hours

Storage instructions

Store at room temperature below 25°C.

Drug interactions

Alcohol; antacids; morphine

Age restrictions

Safe for use in children from 6 years for epilepsy.

Pregnancy and breastfeeding

Use only if the potential benefit outweighs the risk to the foetus.

Precautions and warnings

may cause drowsiness; do not stop treatment abruptly; avoid driving or operating machinery if dizziness occurs

Serious side effects

respiratory depression — requires immediate medical attention; suicidal ideation — requires immediate medical attention; anaphylaxis — requires immediate medical attention

Patient summary

Intended to alleviate chronic neuropathic pain and prevent seizures, utilized to support neurological stability and enhance quality of life.

Mechanism of action

Gabapentin is a structural analogue of the neurotransmitter GABA, although it does not interact directly with GABA receptors. It binds to the alpha-2-delta subunit of voltage-gated calcium channels, which modulates the release of excitatory neurotransmitters.

Neurontin

Intended to alleviate chronic neuropathic pain and prevent seizures, utilized to support neurological stability and enhance quality of life.

Editorial Notes

  • Active ingredient(s): Gabapentin
  • Listed indication(s): Epilepsy, Neuropathic Pain

Usually available as

  • 60 tablets - 300 mg223-300-mg-5078
  • 60 tablets - 400 mg223-400-mg-5085
  • 30 tablets - 600 mg223-600-mg-5090