Ezetimibe Tablets

designed to mitigate high cholesterol levels indicated to support cardiovascular function.

Strengths: 10mg

Medicine details

Alternative names

Ezetrol

Therapeutic class

Cholesterol Absorption Inhibitor

Pharmacological class

Cholesterol Absorption Inhibitor

Contraindications

hypersensitivity; active liver disease

Precautions and warnings

monitor liver function enzymes when combined with statins

Minor side effects

fatigue; abdominal pain; diarrhoea

Moderate side effects

myalgia; elevated liver enzymes

Dosage forms

Tablet

Administration route

Oral use

Prescription status

POM

Manufacturer

Merck Sharp & Dohme

Onset Time

2–4 weeks

Duration

24 hours

Storage instructions

Store below 30°C in the original container.

Drug interactions

ciclosporin; warfarin

Age restrictions

Dosage titration monitored by physician in adolescents.

Pregnancy and breastfeeding

Use not recommended without specialist advice.

Serious side effects

rhabdomyolysis — requires immediate medical attention; hepatitis — requires immediate medical attention

Patient summary

designed to mitigate high cholesterol levels indicated to support cardiovascular function.

Mechanism of action

Ezetimibe inhibits cholesterol absorption at the brush border of the small intestine, blocking the Niemann-Pick C1-like 1 (NPC1L1) transporter protein and reducing deliver of cholesterol to the liver.

Ezetimibe Tablets

designed to mitigate high cholesterol levels indicated to support cardiovascular function.

Editorial Notes

  • Active ingredient(s): Ezetimibe
  • Listed indication(s): Hypercholesterolaemia

Available option

  • 90 tablets - 10 mg1381-10-mg-16577