Chlorambucil Tablets

Developed to target malignancy, utilized to manage symptoms of chronic lymphoid conditions.

Strengths: 2 · 5mg

Medicine details

Alternative names

Leukeran

Therapeutic class

Alkylating Agent

Pharmacological class

Nitrogen Mustard

Contraindications

severe bone marrow suppression; hypersensitivity

Precautions and warnings

regular blood counts required; avoid live vaccines

Minor side effects

nausea; fatigue

Moderate side effects

leukopenia; thrombocytopenia

Dosage forms

Tablet

Administration route

Oral use

Prescription status

POM

Manufacturer

Aspen Pharma

Storage instructions

Store in a refrigerator (2°C–8°C).

Drug interactions

immunosuppressants

Pregnancy and breastfeeding

Pregnancy: Do not use. Breastfeeding: Do not use.

Serious side effects

bone marrow failure — requires immediate medical attention; secondary malignancy — requires immediate medical attention

Patient summary

Developed to target malignancy, utilized to manage symptoms of chronic lymphoid conditions.

Mechanism of action

Chlorambucil is a bifunctional alkylating agent that creates cross-links between DNA strands, inhibiting DNA replication and transcription, which prevents rapidly dividing cancer cells from proliferating.

Chlorambucil Tablets

Developed to target malignancy, utilized to manage symptoms of chronic lymphoid conditions.

Editorial Notes

  • Active ingredient(s): Chlorambucil
  • Listed indication(s): Chronic Lymphocytic Leukaemia, Non-hodgkin Lymphoma

Usually available as

  • 30 tablets - 2 mg1180-2-mg-13962
  • 30 tablets - 5 mg1180-5-mg-13967