Alkacel

Formulated to address malignant cell proliferation by supporting the alkylation of DNA and inhibiting cellular replication.

Strengths: 2mg

Medicine details

Alternative names

Alkeran

Therapeutic class

Antineoplastic Agent; Alkylating Agent

Pharmacological class

Nitrogen Mustard

Contraindications

hypersensitivity to melphalan; severe bone marrow suppression

Minor side effects

nausea; vomiting; alopecia

Moderate side effects

anaemia; leukopenia; thrombocytopenia; stomatitis

Dosage forms

Film-coated tablet

Administration route

Oral use

Prescription status

POM

Manufacturer

Celon Laboratories

Onset Time

N/A

Duration

N/A

Storage instructions

Store at 2–8°C.

Drug interactions

ciclosporin; nalidixic acid

Age restrictions

Use with caution in children.

Pregnancy and breastfeeding

Pregnancy: Contraindicated. Breastfeeding: Contraindicated.

Precautions and warnings

regular blood monitoring recommended; avoid conception during treatment; risk of secondary malignancy

Serious side effects

bone marrow failure — requires immediate medical attention; pulmonary fibrosis — requires immediate medical attention

Patient summary

Formulated to address malignant cell proliferation by supporting the alkylation of DNA and inhibiting cellular replication.

Mechanism of action

Melphalan is a bifunctional alkylating agent that creates cross-links in DNA strands, which interferes with DNA replication and transcription, ultimately inducing apoptosis in malignant cells.

Alkacel

Formulated to address malignant cell proliferation by supporting the alkylation of DNA and inhibiting cellular replication.

Editorial Notes

  • Active ingredient(s): Melphalan
  • Listed indication(s): Multiple Myeloma, Ovarian Cancer

Available option

  • 25 tablets - 2 mg1024-2-mg-12849