Ziprasidone Capsules
Utilized for schizophrenia to alleviate symptoms.
Strengths: 20 · 40 · 80mg
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Medicine details
- Conditions
- Alternative names
Zeldox
- Therapeutic class
Second-Generation Antipsychotic
- Pharmacological class
Atypical Antipsychotic
- Minor side effects
dizziness; somnolence; nausea; dry mouth
- Moderate side effects
constipation; dyspepsia; tachycardia; insomnia
- Dosage forms
Capsule, hard
- Administration route
Oral use
- Patient summary
Utilized for schizophrenia to alleviate symptoms.
- Prescription status
POM
- Manufacturer
Pfizer
- Onset Time
1–2 weeks
- Duration
12–24 hours
- Storage instructions
Store below 30°C in a dry place.
- Drug interactions
QT-prolonging drugs; antiarrhythmics; carbamazepine
- Age restrictions
Not recommended for children under 18.
Contraindications
hypersensitivity to ziprasidone; prolonged QT interval; recent myocardial infarction; uncompensated heart failure
Precautions and warnings
monitor electrocardiogram during treatment; avoid in patients with electrolyte imbalances; may cause drowsiness; regular blood pressure monitoring recommended
Serious side effects
torsades de pointes — requires immediate medical attention; neuroleptic malignant syndrome — requires immediate medical attention
Mechanism of action
Ziprasidone acts as an antagonist at dopamine D2 and serotonin 5-HT2 and 5-HT1 receptors. By modulating these neurotransmitter pathways, it helps balance brain chemical activity, reducing symptoms of psychosis and stabilizing mood in patients with bipolar disorders.
Pregnancy and breastfeeding
Pregnancy: Use only if the potential benefit outweighs the risk. Breastfeeding: Consult a physician as excretion in breast milk is likely.
Ziprasidone Capsules
Utilized for schizophrenia to alleviate symptoms.
Editorial Notes
- Active ingredient(s): Ziprasidone
- Listed indication(s): Schizophrenia, Bipolar Disorder
Usually available as
- 120 tablets - 20 mg1315-20-mg-15717
- 90 tablets - 40 mg1315-40-mg-15705
- 60 tablets - 80 mg1315-80-mg-15710