Warfarin Tablets

Formulated for thromboembolism to mitigate clotting risks.

Strengths: 1 · 2 · 5mg

Medicine details

Alternative names

Marevan; Warfant

Therapeutic class

Vitamin K Antagonist

Pharmacological class

Coumarin Anticoagulant

Minor side effects

bruising; minor bleeding

Moderate side effects

epistaxis; haematuria; alopecia

Dosage forms

Tablet

Administration route

Oral use

Patient summary

Formulated for thromboembolism to mitigate clotting risks.

Prescription status

POM

Manufacturer

Teva UK

Onset Time

48–72 hours

Duration

2–5 days

Storage instructions

Store below 25°C in a dry place.

Drug interactions

Alcohol; Cranberry juice; NSAIDs; Antibiotics

Age restrictions

Use with caution in elderly patients.

Contraindications

pregnancy; severe hypertension; hemorrhagic conditions; severe hepatic impairment

Precautions and warnings

regular blood monitoring required; avoid rapid dietary changes in vitamin k intake; inform your doctor before any planned surgery

Serious side effects

major haemorrhage — requires immediate medical attention; calciphylaxis — requires immediate medical attention

Mechanism of action

Warfarin acts as a vitamin K antagonist by inhibiting the enzyme vitamin K epoxide reductase. This impairs the synthesis of vitamin K-dependent clotting factors II, VII, IX, and X, effectively prolonging the time required for blood to clot.

Pregnancy and breastfeeding

Pregnancy: Contraindicated as it may cause congenital malformations. Breastfeeding: Generally considered safe.

Warfarin Tablets

Formulated for thromboembolism to mitigate clotting risks.

Editorial Notes

  • Active ingredient(s): Warfarin
  • Listed indication(s): Atrial Fibrillation, Thromboembolism, Deep Vein Thrombosis

Usually available as

  • 360 tablets - 1 mg1316-1-mg-15725
  • 360 tablets - 2 mg1316-2-mg-15731
  • 180 tablets - 5 mg1316-5-mg-15738