Protopic

Designed to alleviate atopic dermatitis symptoms, formulated to target skin inflammation and to support to manage flare-ups.

Strengths: 0.03 · 0.1%

Medicine details

Alternative names

Prograf; Adoport

Therapeutic class

Calcineurin inhibitor

Pharmacological class

Immunosuppressant

Contraindications

hypersensitivity to tacrolimus; netherton syndrome

Minor side effects

application site burning; pruritus; erythema

Moderate side effects

folliculitis; skin infections; acne

Serious side effects

malignancy — requires immediate medical attention

Dosage forms

Ointment

Administration route

Cutaneous use

Prescription status

POM

Manufacturer

Leo Laboratories

Onset Time

1 week

Duration

As directed by physician

Storage instructions

Store below 25°C.

Age restrictions

Not for children under 2 years.

Precautions and warnings

avoid alcohol consumption during treatment; minimize exposure to natural or artificial sunlight

Patient summary

Designed to alleviate atopic dermatitis symptoms, formulated to target skin inflammation and to support to manage flare-ups.

Mechanism of action

Tacrolimus inhibits calcineurin, a phosphatase involved in T-lymphocyte activation. By preventing calcineurin activity, it suppresses the transcription of proinflammatory cytokines, thereby reducing inflammation and skin lesions.

Pregnancy and breastfeeding

Pregnancy: Monitor closely; use only if benefit justifies risk. Breastfeeding: Use with caution; consult clinical guidance.

Protopic

Designed to alleviate atopic dermatitis symptoms, formulated to target skin inflammation and to support to manage flare-ups.

Editorial Notes

  • Active ingredient(s): Tacrolimus
  • Listed indication(s): Atopic Dermatitis

Available option

  • 3 tubes - 0.1 %1196-0-1-pct-14168